Pri 35 bolnikih, ki so prejemali 600 mg efavirenza enkrat na dan, so bile v stanju dinamičnega ravnovesja vrednosti Cmax 12, 9 ± 3, 7 µM (29 %) [ povprečje ± standardna deviacija (S. D.) (koeficient variabilnosti (% C. V.)) ], Cmin 5, 6 ± 3, 2 µM (57 %) in AUC 184 ± 73 µM• h (40 %).
In 35 patients receiving efavirenz 600 mg once daily, steady-state peak concentration (Cmax) was 12.9 ± 3.7 µM (29 %) [ mean ± standard deviation (S. D.) (coefficient of variation (%CV)) ], steady-state Cmin was 5.6 ± 3.2 µM (57 %), and AUC was 184 ± 73 µM• h (40 %).